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As carisoprodol and its metabolite meprobamate are GABA receptor agonists, the use of the benzodiazepine receptor antagonist flumazenil might be considered in some cases of carisoprodol toxicity. The Drug Enforcement Administration lists the following physical effects: Agitation. Irritability. Depression. Carisoprodol is an FDA-approved drug indicated for the relief of discomfort associated with acute, painful musculoskeletal conditions. It has approval for up to three weeks of use only.
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